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Competitive inhibition of calcineurin phosphatase activity by its autoinhibitory domain.

Calcineurin (protein phosphatase 2B), a calmodulin- and calcium-dependent serine/threonine phosphatase, appears to be regulated by a C-terminal autoinhibitory domain. A 25 amino acid peptide derived from this domain inhibits calcineurin phosphatase activity in vitro. Here we show that a 97 amino aci...

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Detalhes bibliográficos
Main Authors: Sagoo, J K, Fruman, D A, Wesselborg, S, Walsh, C T, Bierer, B E
Formato: Artigo
Idioma:Inglês
Publicado em: 1996
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC1218010/
https://ncbi.nlm.nih.gov/pubmed/9003375
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