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Expanded Physiologically‐Based Pharmacokinetic Model of Rifampicin for Predicting Interactions With Drugs and an Endogenous Biomarker via Complex Mechanisms Including Organic Anion Transporting Polypeptide 1B Induction

As rifampicin can cause the induction and inhibition of multiple metabolizing enzymes and transporters, it has been challenging to accurately predict the complex drug–drug interactions (DDIs). We previously constructed a physiologically‐based pharmacokinetic (PBPK) model of rifampicin accounting for...

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Xehetasun bibliografikoak
Egile Nagusiak: Ryuta Asaumi, Karsten Menzel, Wooin Lee, Ken‐ichi Nunoya, Haruo Imawaka, Hiroyuki Kusuhara, Yuichi Sugiyama
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Wiley 2019-11-01
Saila:CPT: Pharmacometrics & Systems Pharmacology
Sarrera elektronikoa:https://doi.org/10.1002/psp4.12457
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