Cinchona Alkaloid Derivative-Catalyzed Enantioselective Synthesis via a Mannich-Type Reaction and Antifungal Activity of β-Amino Esters Bearing Benzoheterocycle Moieties

An efficient synthesis of highly functionalized chiral β-amino ester derivatives containing benzothiophene and benzothiazole moieties is developed by a Mannich-type reaction using a cinchona alkaloid-derived thiourea catalyst. The desired products were obtained in good yields and high enantioselecti...

Descripción completa

Guardado en:
Detalles Bibliográficos
Autores principales: Han Xiao, Fang Wu, Li Shi, Zhiwei Chen, Shihu Su, Chenghao Tang, Hongtao Wang, Zhining Li, Meichuan Li, Qingcai Shi
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI AG 2014-04-01
Colección:Molecules
Materias:
β-amino acid ester
antifungal activity
benzoheterocycle
enantioselective synthesis
Acceso en línea:http://www.mdpi.com/1420-3049/19/4/3955
Etiquetas: Agregar Etiqueta
Sin Etiquetas, Sea el primero en etiquetar este registro!

Ejemplares similares