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Selective DNA Gyrase Inhibitors: Multi-Target in Silico Profiling with 3D-Pharmacophores

DNA gyrase is an important target for the development of novel antibiotics. Although ATP-competitive DNA gyrase (GyrB) inhibitors are a well-studied class of antibacterial agents, there is currently no representative used in therapy, largely due to unwanted off-target activities. Selectivity of GyrB...

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Furkejuvvon:
Bibliográfalaš dieđut
Váldodahkkit: Tihomir Tomašič, Asta Zubrienė, Žiga Skok, Riccardo Martini, Stane Pajk, Izidor Sosič, Janez Ilaš, Daumantas Matulis, Sharon D. Bryant
Materiálatiipa: Artigo
Giella:Inglês
Almmustuhtton: MDPI AG 2021-08-01
Ráidu:Pharmaceuticals
Fáttát:
Liŋkkat:https://www.mdpi.com/1424-8247/14/8/789
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