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Conformational dynamics of a nicotinic receptor neurotransmitter site

Agonists enhance receptor activity by providing net-favorable binding energy to active over resting conformations, with efficiency (η) linking binding energy to gating. Previously, we showed that in nicotinic receptors, η-values are grouped into five structural pairs, correlating efficacy and affini...

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Autori principali: Mrityunjay Singh, Dinesh C Indurthi, Lovika Mittal, Anthony Auerbach, Shailendra Asthana
Natura: Artigo
Lingua:Inglês
Pubblicazione: eLife Sciences Publications Ltd 2024-12-01
Serie:eLife
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Accesso online:https://elifesciences.org/articles/92418
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