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Intracellular pharmacokinetic study of zidovudine and its phosphorylated metabolites

Zidovudine (AZT), the first drug approved by the US Food and Drug Administration for the treatment of human immunodeficiency virus (HIV) infection, is metabolized in the host cells to 5′-AZT triphosphate (AZT-TP) which inhibits HIV reverse transcriptase. As the pharmacokinetics of AZT and its phosph...

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-д хадгалсан:
Номзүйн дэлгэрэнгүй
Үндсэн зохиолчид: Lingli Mu, Rui Zhou, Fang Tang, Xingling Liu, Sanwang Li, Feifan Xie, Xiang Xie, Jie Peng, Peng Yu
Формат: Artigo
Хэл сонгох:Inglês
Хэвлэсэн: Elsevier 2016-03-01
Цуврал:Acta Pharmaceutica Sinica B
Нөхцлүүд:
Онлайн хандалт:http://www.sciencedirect.com/science/article/pii/S2211383515001434
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