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SUMOylation inhibitors synergize with FXR agonists in combating liver fibrosis

Abstract Farnesoid X receptor (FXR) is a promising target for nonalcoholic steatohepatitis (NASH) and fibrosis. Although various FXR agonists have shown anti-fibrotic effects in diverse preclinical animal models, the response rate and efficacies in clinical trials were not optimum. Here we report th...

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Autors principals: Jiyu Zhou, Shuang Cui, Qingxian He, Yitong Guo, Xiaojie Pan, Pengfei Zhang, Ningning Huang, Chaoliang Ge, Guangji Wang, Frank J. Gonzalez, Hong Wang, Haiping Hao
Format: Artigo
Idioma:Inglês
Publicat: Nature Portfolio 2020-01-01
Col·lecció:Nature Communications
Accés en línia:https://doi.org/10.1038/s41467-019-14138-6
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