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Effects of Cyclization on Activity and Stability of α-Conotoxin TxIB

α-Conotoxin TxIB specifically blocked α6/α3β2β3 acetylcholine receptors (nAChRs), and it could be a potential probe for studying addiction and other diseases related to α6/α3β2β3 nAChRs. However, as a peptide, TxIB may suffer from low stability, short half-life, and poor bioavailability. In this stu...

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Principais autores: Xincan Li, Shuai Wang, Xiaopeng Zhu, Dongting Zhangsun, Yong Wu, Sulan Luo
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI AG 2020-03-01
Colecção:Marine Drugs
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Acesso em linha:https://www.mdpi.com/1660-3397/18/4/180
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