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Safety, Tolerability, and Pharmacokinetics of KP-1461 in Phase I Clinical Studies

Background: KP-1461 is a prodrug to KP-1212. KP-1212 is a viral mutagen designed to increase viral error rate. Methods: We describe 2 phase I studies: KP1461-101 (double-blind, placebo-controlled, single, escalating doses, 100 to 1600 mg study in 42 non-HIV-infected participants) and KP-1461-102 (do...

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Principais autores: Patrick G. Clay PharmD, MaryPeace McRae PharmD, PhD, Jean-Pierre Laurent
Formato: Artigo
Idioma:Inglês
Publicado: SAGE Publishing 2011-08-01
Series:Journal of the International Association of Providers of AIDS Care
Acceso en liña:https://doi.org/10.1177/1545109711406442
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