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Synthesis of Berberine and Canagliflozin Chimera and Investigation into New Antibacterial Activity and Mechanisms

Berberine is an isoquinoline alkaloid isolated from Chinese herbal medicines such as Coptis chinensis. It has many pharmacological actions, such as antibacterial, hypoglycemic, anti-inflammatory, and so on. However, due to the low lipophilicity of berberine, it is difficult to penetrate the bacteria...

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Principais autores: Wenhui Hao, Shiying Che, Jinsheng Li, Jingyi Luo, Wanqiu Zhang, Yang Chen, Zijian Zhao, Hao Wei, Weidong Xie
Formato: Artigo
Idioma:Inglês
Publicado: MDPI AG 2022-05-01
Series:Molecules
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Acceso en liña:https://www.mdpi.com/1420-3049/27/9/2948
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