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Design and Synthesis of 2,6-Disubstituted-4′-Selenoadenosine-5′-<em>N</em>,<em>N</em>-Dimethyluronamide Derivatives as Human A<sub>3</sub> Adenosine Receptor Antagonists

A new series of 4′-selenoadenosine-5′-<i>N,N</i>-dimethyluronamide derivatives as highly potent and selective human A<sub>3</sub> adenosine receptor (hA<sub>3</sub>AR) antagonists, is described. The highly selective A<sub>3</sub>AR agonists, 4′-selenoadenosine-5′-<i>N</i>-methyluronamides were succe...

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Autors principals: Hongseok Choi, Kenneth A. Jacobson, Jinha Yu, Lak Shin Jeong
Format: Artigo
Idioma:Inglês
Publicat: MDPI AG 2021-04-01
Col·lecció:Pharmaceuticals
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Accés en línia:https://www.mdpi.com/1424-8247/14/4/363
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