Design and Synthesis of 2,6-Disubstituted-4′-Selenoadenosine-5′-<em>N</em>,<em>N</em>-Dimethyluronamide Derivatives as Human A<sub>3</sub> Adenosine Receptor Antagonists
A new series of 4′-selenoadenosine-5′-<i>N,N</i>-dimethyluronamide derivatives as highly potent and selective human A<sub>3</sub> adenosine receptor (hA<sub>3</sub>AR) antagonists, is described. The highly selective A<sub>3</sub>AR agonists, 4′-selenoadenosine-5′-<i>N</i>-methyluronamides were succe...
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| Autors principals: | , , , |
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| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
MDPI AG
2021-04-01
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| Col·lecció: | Pharmaceuticals |
| Matèries: | |
| Accés en línia: | https://www.mdpi.com/1424-8247/14/4/363 |
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