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Molecular basis for depsipeptide HDAC inhibitor combinatorial biosynthesis

Abstract Polyketides and nonribosomal peptides are important natural product classes with wide-ranging medical and agricultural applications. The analogous enzymatic logic employed by bacterial modular polyketide synthases (PKSs) and nonribosomal peptide synthetases (NRPSs) enables the assembly of h...

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Egile Nagusiak: Munro Passmore, Xinyun Jian, Xinyi Zhao, Emmanuel L. C. de los Santos, Douglas M. Roberts, Józef R. Lewandowski, Matthew Jenner, Lona M. Alkhalaf, Gregory L. Challis
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Nature Portfolio 2026-07-01
Saila:Nature Communications
Sarrera elektronikoa:https://doi.org/10.1038/s41467-026-74383-4
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