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New Uncharged 2-Thienostilbene Oximes as Reactivators of Organophosphate-Inhibited Cholinesterases

The inhibition of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE) by organophosphates (OPs) as nerve agents and pesticides compromises normal cholinergic nerve signal transduction in the peripheral and central nervous systems (CNS) leading to cholinergic crisis. The treatment comprises...

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Hlavní autoři: Milena Mlakić, Tena Čadež, Danijela Barić, Ivana Puček, Ana Ratković, Željko Marinić, Kornelija Lasić, Zrinka Kovarik, Irena Škorić
Médium: Artigo
Jazyk:Inglês
Vydáno: MDPI AG 2021-11-01
Edice:Pharmaceuticals
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On-line přístup:https://www.mdpi.com/1424-8247/14/11/1147
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