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Pathophysiological Role and Medicinal Chemistry of A<sub>2A</sub> Adenosine Receptor Antagonists in Alzheimer’s Disease

The A<sub>2A</sub> adenosine receptor is a protein belonging to a family of four GPCR adenosine receptors. It is involved in the regulation of several pathophysiological conditions in both the central nervous system and periphery. In the brain, its localization at pre- and postsynaptic level in stri...

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Autores principales: Stefania Merighi, Pier Andrea Borea, Katia Varani, Fabrizio Vincenzi, Alessia Travagli, Manuela Nigro, Silvia Pasquini, R. Rama Suresh, Sung Won Kim, Nora D. Volkow, Kenneth A. Jacobson, Stefania Gessi
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI AG 2022-04-01
Colección:Molecules
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Acceso en línea:https://www.mdpi.com/1420-3049/27/9/2680
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