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Novel inhibitors of phosphorylation independent activity of GRK2 modulate cAMP signaling

Abstract G protein‐coupled receptors kinase 2 (GRK2) plays a major role in receptor regulation and, as a consequence, in cell biology and physiology. GRK2‐mediated receptor desensitization is performed by its kinase domain, which exerts receptor phosphorylation promoting G protein uncoupling and the...

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Hlavní autoři: Emiliana Echeverría, Sonia Ripoll, Lucas Fabián, Carina Shayo, Federico Monczor, Natalia C. Fernández
Médium: Artigo
Jazyk:Inglês
Vydáno: Wiley 2022-04-01
Edice:Pharmacology Research & Perspectives
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On-line přístup:https://doi.org/10.1002/prp2.913
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