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Characterization of Stimulatory Action on Voltage-Gated Na<sup>+</sup> Currents Caused by Omecamtiv Mecarbil, Known to Be a Myosin Activator

Omecamtiv mecarbil (OM, CK-1827452) is recognized as an activator of myosin and has been demonstrated to be beneficial for the treatment of systolic heart failure. However, the mechanisms by which this compound interacts with ionic currents in electrically excitable cells remain largely unknown. The...

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Xehetasun bibliografikoak
Egile Nagusiak: Chih-Yu Ting, Chia-Lung Shih, Meng-Cheng Yu, Chao-Liang Wu, Sheng-Nan Wu
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: MDPI AG 2023-05-01
Saila:Biomedicines
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Sarrera elektronikoa:https://www.mdpi.com/2227-9059/11/5/1351
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