Modulation of K(v)11.1 (hERG) channels by 5‐(((1H–indazol‐5‐yl)oxy)methyl)‐N‐(4‐(trifluoromethoxy)phenyl)pyrimidin‐2‐amine (ITP‐2), a novel small molecule activator...

Por Sale, Harinath, Roy, Samrat, Warrier, Jayakumar, Thangathirupathy, Srinivasan, Vadari, Yoganand, Gopal, Shruthi K, Krishnamurthy, Prasad, Ramarao, Manjunath
Publicado no Br J Pharmacol (2017)

BMS-986163, a Negative Allosteric Modulator of GluN2B with Potential Utility in Major Depressive Disorder

Por Marcin, Lawrence R., Warrier, Jayakumar, Thangathirupathy, Srinivasan, Shi, Jianliang, Karageorge, George N., Pearce, Bradley C., Ng, Alicia, Park, Hyunsoo, Kempson, James, Li, Jianqing, Zhang, Huiping, Mathur, Arvind, Reddy, Aliphedi B., Nagaraju, G., Tonukunuru, Gopikishan, Gupta, Grandhi V. R. K. M., Kamble, Manjunatha, Mannoori, Raju, Cheruku, Srinivas, Jogi, Srinivas, Gulia, Jyoti, Bastia, Tanmaya, Sanmathi, Charulatha, Aher, Jayant, Kallem, Rajareddy, Srikumar, Bettadapura N., Vijaya, Kumar Kuchibhotla, Naidu, Pattipati S., Paschapur, Mahesh, Kalidindi, Narasimharaju, Vikramadithyan, Reeba, Ramarao, Manjunath, Denton, Rex, Molski, Thaddeus, Shields, Eric, Subramanian, Murali, Zhuo, Xiaoliang, Nophsker, Michelle, Simmermacher, Jean, Sinz, Michael, Albright, Charlie, Bristow, Linda J., Islam, Imadul, Bronson, Joanne J., Olson, Richard E., King, Dalton, Thompson, Lorin A., Macor, John E.
Publicado no ACS Med Chem Lett (2018)