Structure-Based Design of Irreversible Human KAT II Inhibitors: Discovery of New Potency-Enhancing Interactions

por Tuttle, Jamison B., Anderson, Marie, Bechle, Bruce M., Campbell, Brian M., Chang, Cheng, Dounay, Amy B., Evrard, Edelweiss, Fonseca, Kari R., Gan, Xinmin, Ghosh, Somraj, Horner, Weldon, James, Larry C., Kim, Ji-Young, McAllister, Laura A., Pandit, Jayvardhan, Parikh, Vinod D., Rago, Brian J., Salafia, Michelle A., Strick, Christine A., Zawadzke, Laura E., Verhoest, Patrick R.
Publicado 2012

Discovery of Brain-Penetrant, Irreversible Kynurenine Aminotransferase II Inhibitors for Schizophrenia

por Dounay, Amy B., Anderson, Marie, Bechle, Bruce M., Campbell, Brian M., Claffey, Michelle M., Evdokimov, Artem, Evrard, Edelweiss, Fonseca, Kari R., Gan, Xinmin, Ghosh, Somraj, Hayward, Matthew M., Horner, Weldon, Kim, Ji-Young, McAllister, Laura A., Pandit, Jayvardhan, Paradis, Vanessa, Parikh, Vinod D., Reese, Matthew R., Rong, SuoBao, Salafia, Michelle A., Schuyten, Katherine, Strick, Christine A., Tuttle, Jamison B., Valentine, James, Wang, Hong, Zawadzke, Laura E., Verhoest, Patrick R.
Publicado 2012