A General Protocol for Cu-Mediated Fluoro-deamination: Sandmeyer Fluorination of Diverse Aromatic Substrates

Yazar: Pérez-García, R. Manuel, Grønnevik, Gaute, Riss, Patrick J.
Yayımlandı Org Lett (2021)

Synthesis and Characterization in Rodent Brain of the Subtype-Selective NR2B NMDA Receptor Ligand [(11)C]Ro04-5595 as a Potential Radiotracer for Positron Emission Tomography

Yazar: Jakobsson, Jimmy E., Gourni, Eleni, Khanapur, Shivashankar, Brito, Beatriz, Riss, Patrick J.
Yayımlandı ACS Omega (2019)

Cu(I)-catalyzed (11)C-carboxylation of boronic acid esters: a rapid and convenient entry to (11)C-labeled carboxylic acids, esters and amides

Yazar: Riss, Patrick J., Lu, Shuiyu, Telu, Sanjay, Aigbirhio, Franklin I., Pike, Victor W.
Baskı/Yayın Bilgisi 2012

Small molecule piperazinyl-benzimidazole antagonists of the gonadotropin-releasing hormone (GnRH) receptor

Yazar: Fjellaksel, Richard, Boomgaren, Marc, Sundset, Rune, Haraldsen, Ira H., Hansen, Jørn H., Riss, Patrick J.
Yayımlandı Medchemcomm (2017)

Recent Development of Non-Peptide GnRH Antagonists

Yazar: Tukun, Feng-Ling, Olberg, Dag Erlend, Riss, Patrick J., Haraldsen, Ira, Kaass, Anita, Klaveness, Jo
Yayımlandı Molecules (2017)

Radiosynthesis and validation of (18)F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain

Yazar: Cumming, Paul, Maschauer, Simone, Riss, Patrick J, Tschammer, Nuska, Fehler, Stefanie K, Heinrich, Markus R, Kuwert, Torsten, Prante, Olaf
Baskı/Yayın Bilgisi 2014

First in vivo evaluation of a potential SPECT brain radiotracer for the gonadotropin releasing hormone receptor

Yazar: Fjellaksel, Richard, Oteiza, Ana, Martin-Armas, Montserrat, Riss, Patrick J., Hjelstuen, Ole Kristian, Kuttner, Samuel, Hansen, Jørn H., Sundset, Rune
Yayımlandı BMC Res Notes (2018)

[(18)F]PR04.MZ PET/CT Imaging for Evaluation of Nigrostriatal Neuron Integrity in Patients With Parkinson Disease

Yazar: Juri, Carlos, Kramer, Vasko, Riss, Patrick J., Soza-Ried, Cristian, Haeger, Arlette, Pruzzo, Rossana, Rösch, Frank, Amaral, Horacio, Chana-Cuevas, Pedro
Yayımlandı Clin Nucl Med (2021)

Pharmacological Characterization of Low-to-Moderate Affinity Opioid Receptor Agonists and Brain Imaging with (18)F-Labeled Derivatives in Rats

Yazar: Ott, Julian, Spilhaug, Mona M., Maschauer, Simone, Rafique, Waqas, Jakobsson, Jimmy E., Hartvig, Karoline, Hübner, Harald, Gmeiner, Peter, Prante, Olaf, Riss, Patrick J.
Yayımlandı J Med Chem (2020)

Discovery of a Lead Brain‐Penetrating Gonadotropin‐Releasing Hormone Receptor Antagonist with Saturable Binding in Brain

Yazar: Bekker, Roberto B. W., Fjellaksel, Richard, Hjornevik, Trine, Nuruddin, Syed, Rafique, Waqas, Hansen, Jørn H., Sundset, Rune, Haraldsen, Ira H., Riss, Patrick J.
Yayımlandı ChemMedChem (2020)

Image-Guided Development of Heterocyclic Sulfoxides as Ligands for Tau Neurofibrillary Tangles: From First-in-Man to Second-Generation Ligands

Yazar: Rafique, Waqas, Kramer, Vasko, Pardo, Tania, Smits, René, Spilhaug, Mona M., Hoepping, Alexander, Savio, Eduardo, Engler, Henry, Kuljs, Rodrigo, Amaral, Horacio, Riss, Patrick J.
Yayımlandı ACS Omega (2018)

Validation and quantification of [(18)F]altanserin binding in the rat brain using blood input and reference tissue modeling

Yazar: Riss, Patrick J, Hong, Young T, Williamson, David, Caprioli, Daniele, Sitnikov, Sergey, Ferrari, Valentina, Sawiak, Steve J, Baron, Jean-Claude, Dalley, Jeffrey W, Fryer, Tim D, Aigbirhio, Franklin I
Baskı/Yayın Bilgisi 2011

Evaluation of [(18)F]N-methyl-lansoprazole as a tau PET imaging agent in first-in-human studies

Yazar: Kramer, Vasko, Brooks, Allen F., Haeger, Arlette, Kuljis, Rodrigo, Rafique, Waqas, Koeppe, Robert A., Raffel, David M., Frey, Kirk A., Amaral, Horacio, Scott, Peter J. H., Riss, Patrick J.
Yayımlandı ACS Chem Neurosci (2020)

Insula serotonin 2A receptor binding and gene expression contribute to serotonin transporter polymorphism anxious phenotype in primates

Yazar: Santangelo, Andrea M., Sawiak, Steve J., Fryer, Tim, Hong, Young, Shiba, Yoshiro, Clarke, Hannah F., Riss, Patrick J., Ferrari, Valentina, Tait, Roger, Suckling, John, Aigbirhio, Franklin I., Roberts, Angela C.
Yayımlandı Proc Natl Acad Sci U S A (2019)

Synthesis and Initial in Vivo Studies with [(11)C]SB-216763: The First Radiolabeled Brain Penetrative Inhibitor of GSK-3

Yazar: Li, Lei, Shao, Xia, Cole, Erin L., Ohnmacht, Stephan A., Ferrari, Valentina, Hong, Young T., Williamson, David J., Fryer, Tim D., Quesada, Carole A., Sherman, Phillip, Riss, Patrick J., Scott, Peter J. H., Aigbirhio, Franklin I.
Yayımlandı ACS Med Chem Lett (2015)