A General Protocol for Cu-Mediated Fluoro-deamination: Sandmeyer Fluorination of Diverse Aromatic Substrates

door Pérez-García, R. Manuel, Grønnevik, Gaute, Riss, Patrick J.
Gepubliceerd in Org Lett (2021)

Synthesis and Characterization in Rodent Brain of the Subtype-Selective NR2B NMDA Receptor Ligand [(11)C]Ro04-5595 as a Potential Radiotracer for Positron Emission Tomography

door Jakobsson, Jimmy E., Gourni, Eleni, Khanapur, Shivashankar, Brito, Beatriz, Riss, Patrick J.
Gepubliceerd in ACS Omega (2019)

Cu(I)-catalyzed (11)C-carboxylation of boronic acid esters: a rapid and convenient entry to (11)C-labeled carboxylic acids, esters and amides

door Riss, Patrick J., Lu, Shuiyu, Telu, Sanjay, Aigbirhio, Franklin I., Pike, Victor W.
Gepubliceerd in 2012

Small molecule piperazinyl-benzimidazole antagonists of the gonadotropin-releasing hormone (GnRH) receptor

door Fjellaksel, Richard, Boomgaren, Marc, Sundset, Rune, Haraldsen, Ira H., Hansen, Jørn H., Riss, Patrick J.
Gepubliceerd in Medchemcomm (2017)

Recent Development of Non-Peptide GnRH Antagonists

door Tukun, Feng-Ling, Olberg, Dag Erlend, Riss, Patrick J., Haraldsen, Ira, Kaass, Anita, Klaveness, Jo
Gepubliceerd in Molecules (2017)

Radiosynthesis and validation of (18)F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain

door Cumming, Paul, Maschauer, Simone, Riss, Patrick J, Tschammer, Nuska, Fehler, Stefanie K, Heinrich, Markus R, Kuwert, Torsten, Prante, Olaf
Gepubliceerd in 2014

First in vivo evaluation of a potential SPECT brain radiotracer for the gonadotropin releasing hormone receptor

door Fjellaksel, Richard, Oteiza, Ana, Martin-Armas, Montserrat, Riss, Patrick J., Hjelstuen, Ole Kristian, Kuttner, Samuel, Hansen, Jørn H., Sundset, Rune
Gepubliceerd in BMC Res Notes (2018)

[(18)F]PR04.MZ PET/CT Imaging for Evaluation of Nigrostriatal Neuron Integrity in Patients With Parkinson Disease

door Juri, Carlos, Kramer, Vasko, Riss, Patrick J., Soza-Ried, Cristian, Haeger, Arlette, Pruzzo, Rossana, Rösch, Frank, Amaral, Horacio, Chana-Cuevas, Pedro
Gepubliceerd in Clin Nucl Med (2021)

Pharmacological Characterization of Low-to-Moderate Affinity Opioid Receptor Agonists and Brain Imaging with (18)F-Labeled Derivatives in Rats

door Ott, Julian, Spilhaug, Mona M., Maschauer, Simone, Rafique, Waqas, Jakobsson, Jimmy E., Hartvig, Karoline, Hübner, Harald, Gmeiner, Peter, Prante, Olaf, Riss, Patrick J.
Gepubliceerd in J Med Chem (2020)

Discovery of a Lead Brain‐Penetrating Gonadotropin‐Releasing Hormone Receptor Antagonist with Saturable Binding in Brain

door Bekker, Roberto B. W., Fjellaksel, Richard, Hjornevik, Trine, Nuruddin, Syed, Rafique, Waqas, Hansen, Jørn H., Sundset, Rune, Haraldsen, Ira H., Riss, Patrick J.
Gepubliceerd in ChemMedChem (2020)

Image-Guided Development of Heterocyclic Sulfoxides as Ligands for Tau Neurofibrillary Tangles: From First-in-Man to Second-Generation Ligands

door Rafique, Waqas, Kramer, Vasko, Pardo, Tania, Smits, René, Spilhaug, Mona M., Hoepping, Alexander, Savio, Eduardo, Engler, Henry, Kuljs, Rodrigo, Amaral, Horacio, Riss, Patrick J.
Gepubliceerd in ACS Omega (2018)

Validation and quantification of [(18)F]altanserin binding in the rat brain using blood input and reference tissue modeling

door Riss, Patrick J, Hong, Young T, Williamson, David, Caprioli, Daniele, Sitnikov, Sergey, Ferrari, Valentina, Sawiak, Steve J, Baron, Jean-Claude, Dalley, Jeffrey W, Fryer, Tim D, Aigbirhio, Franklin I
Gepubliceerd in 2011

Evaluation of [(18)F]N-methyl-lansoprazole as a tau PET imaging agent in first-in-human studies

door Kramer, Vasko, Brooks, Allen F., Haeger, Arlette, Kuljis, Rodrigo, Rafique, Waqas, Koeppe, Robert A., Raffel, David M., Frey, Kirk A., Amaral, Horacio, Scott, Peter J. H., Riss, Patrick J.
Gepubliceerd in ACS Chem Neurosci (2020)

Insula serotonin 2A receptor binding and gene expression contribute to serotonin transporter polymorphism anxious phenotype in primates

door Santangelo, Andrea M., Sawiak, Steve J., Fryer, Tim, Hong, Young, Shiba, Yoshiro, Clarke, Hannah F., Riss, Patrick J., Ferrari, Valentina, Tait, Roger, Suckling, John, Aigbirhio, Franklin I., Roberts, Angela C.
Gepubliceerd in Proc Natl Acad Sci U S A (2019)

Synthesis and Initial in Vivo Studies with [(11)C]SB-216763: The First Radiolabeled Brain Penetrative Inhibitor of GSK-3

door Li, Lei, Shao, Xia, Cole, Erin L., Ohnmacht, Stephan A., Ferrari, Valentina, Hong, Young T., Williamson, David J., Fryer, Tim D., Quesada, Carole A., Sherman, Phillip, Riss, Patrick J., Scott, Peter J. H., Aigbirhio, Franklin I.
Gepubliceerd in ACS Med Chem Lett (2015)