A General Protocol for Cu-Mediated Fluoro-deamination: Sandmeyer Fluorination of Diverse Aromatic Substrates

por Pérez-García, R. Manuel, Grønnevik, Gaute, Riss, Patrick J.
Publicado en Org Lett (2021)

Synthesis and Characterization in Rodent Brain of the Subtype-Selective NR2B NMDA Receptor Ligand [(11)C]Ro04-5595 as a Potential Radiotracer for Positron Emission Tomography

por Jakobsson, Jimmy E., Gourni, Eleni, Khanapur, Shivashankar, Brito, Beatriz, Riss, Patrick J.
Publicado en ACS Omega (2019)

Cu(I)-catalyzed (11)C-carboxylation of boronic acid esters: a rapid and convenient entry to (11)C-labeled carboxylic acids, esters and amides

por Riss, Patrick J., Lu, Shuiyu, Telu, Sanjay, Aigbirhio, Franklin I., Pike, Victor W.
Publicado 2012

Small molecule piperazinyl-benzimidazole antagonists of the gonadotropin-releasing hormone (GnRH) receptor

por Fjellaksel, Richard, Boomgaren, Marc, Sundset, Rune, Haraldsen, Ira H., Hansen, Jørn H., Riss, Patrick J.
Publicado en Medchemcomm (2017)

Recent Development of Non-Peptide GnRH Antagonists

por Tukun, Feng-Ling, Olberg, Dag Erlend, Riss, Patrick J., Haraldsen, Ira, Kaass, Anita, Klaveness, Jo
Publicado en Molecules (2017)

Radiosynthesis and validation of (18)F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain

por Cumming, Paul, Maschauer, Simone, Riss, Patrick J, Tschammer, Nuska, Fehler, Stefanie K, Heinrich, Markus R, Kuwert, Torsten, Prante, Olaf
Publicado 2014

First in vivo evaluation of a potential SPECT brain radiotracer for the gonadotropin releasing hormone receptor

por Fjellaksel, Richard, Oteiza, Ana, Martin-Armas, Montserrat, Riss, Patrick J., Hjelstuen, Ole Kristian, Kuttner, Samuel, Hansen, Jørn H., Sundset, Rune
Publicado en BMC Res Notes (2018)

[(18)F]PR04.MZ PET/CT Imaging for Evaluation of Nigrostriatal Neuron Integrity in Patients With Parkinson Disease

por Juri, Carlos, Kramer, Vasko, Riss, Patrick J., Soza-Ried, Cristian, Haeger, Arlette, Pruzzo, Rossana, Rösch, Frank, Amaral, Horacio, Chana-Cuevas, Pedro
Publicado en Clin Nucl Med (2021)

Pharmacological Characterization of Low-to-Moderate Affinity Opioid Receptor Agonists and Brain Imaging with (18)F-Labeled Derivatives in Rats

por Ott, Julian, Spilhaug, Mona M., Maschauer, Simone, Rafique, Waqas, Jakobsson, Jimmy E., Hartvig, Karoline, Hübner, Harald, Gmeiner, Peter, Prante, Olaf, Riss, Patrick J.
Publicado en J Med Chem (2020)

Discovery of a Lead Brain‐Penetrating Gonadotropin‐Releasing Hormone Receptor Antagonist with Saturable Binding in Brain

por Bekker, Roberto B. W., Fjellaksel, Richard, Hjornevik, Trine, Nuruddin, Syed, Rafique, Waqas, Hansen, Jørn H., Sundset, Rune, Haraldsen, Ira H., Riss, Patrick J.
Publicado en ChemMedChem (2020)

Image-Guided Development of Heterocyclic Sulfoxides as Ligands for Tau Neurofibrillary Tangles: From First-in-Man to Second-Generation Ligands

por Rafique, Waqas, Kramer, Vasko, Pardo, Tania, Smits, René, Spilhaug, Mona M., Hoepping, Alexander, Savio, Eduardo, Engler, Henry, Kuljs, Rodrigo, Amaral, Horacio, Riss, Patrick J.
Publicado en ACS Omega (2018)

Validation and quantification of [(18)F]altanserin binding in the rat brain using blood input and reference tissue modeling

por Riss, Patrick J, Hong, Young T, Williamson, David, Caprioli, Daniele, Sitnikov, Sergey, Ferrari, Valentina, Sawiak, Steve J, Baron, Jean-Claude, Dalley, Jeffrey W, Fryer, Tim D, Aigbirhio, Franklin I
Publicado 2011

Evaluation of [(18)F]N-methyl-lansoprazole as a tau PET imaging agent in first-in-human studies

por Kramer, Vasko, Brooks, Allen F., Haeger, Arlette, Kuljis, Rodrigo, Rafique, Waqas, Koeppe, Robert A., Raffel, David M., Frey, Kirk A., Amaral, Horacio, Scott, Peter J. H., Riss, Patrick J.
Publicado en ACS Chem Neurosci (2020)

Insula serotonin 2A receptor binding and gene expression contribute to serotonin transporter polymorphism anxious phenotype in primates

por Santangelo, Andrea M., Sawiak, Steve J., Fryer, Tim, Hong, Young, Shiba, Yoshiro, Clarke, Hannah F., Riss, Patrick J., Ferrari, Valentina, Tait, Roger, Suckling, John, Aigbirhio, Franklin I., Roberts, Angela C.
Publicado en Proc Natl Acad Sci U S A (2019)

Synthesis and Initial in Vivo Studies with [(11)C]SB-216763: The First Radiolabeled Brain Penetrative Inhibitor of GSK-3

por Li, Lei, Shao, Xia, Cole, Erin L., Ohnmacht, Stephan A., Ferrari, Valentina, Hong, Young T., Williamson, David J., Fryer, Tim D., Quesada, Carole A., Sherman, Phillip, Riss, Patrick J., Scott, Peter J. H., Aigbirhio, Franklin I.
Publicado en ACS Med Chem Lett (2015)