A General Protocol for Cu-Mediated Fluoro-deamination: Sandmeyer Fluorination of Diverse Aromatic Substrates

ανά Pérez-García, R. Manuel, Grønnevik, Gaute, Riss, Patrick J.
Τόπος έκδοσης Org Lett (2021)

Synthesis and Characterization in Rodent Brain of the Subtype-Selective NR2B NMDA Receptor Ligand [(11)C]Ro04-5595 as a Potential Radiotracer for Positron Emission Tomography

ανά Jakobsson, Jimmy E., Gourni, Eleni, Khanapur, Shivashankar, Brito, Beatriz, Riss, Patrick J.
Τόπος έκδοσης ACS Omega (2019)

Cu(I)-catalyzed (11)C-carboxylation of boronic acid esters: a rapid and convenient entry to (11)C-labeled carboxylic acids, esters and amides

ανά Riss, Patrick J., Lu, Shuiyu, Telu, Sanjay, Aigbirhio, Franklin I., Pike, Victor W.
Έκδοση 2012

Small molecule piperazinyl-benzimidazole antagonists of the gonadotropin-releasing hormone (GnRH) receptor

ανά Fjellaksel, Richard, Boomgaren, Marc, Sundset, Rune, Haraldsen, Ira H., Hansen, Jørn H., Riss, Patrick J.
Τόπος έκδοσης Medchemcomm (2017)

Recent Development of Non-Peptide GnRH Antagonists

ανά Tukun, Feng-Ling, Olberg, Dag Erlend, Riss, Patrick J., Haraldsen, Ira, Kaass, Anita, Klaveness, Jo
Τόπος έκδοσης Molecules (2017)

Radiosynthesis and validation of (18)F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain

ανά Cumming, Paul, Maschauer, Simone, Riss, Patrick J, Tschammer, Nuska, Fehler, Stefanie K, Heinrich, Markus R, Kuwert, Torsten, Prante, Olaf
Έκδοση 2014

First in vivo evaluation of a potential SPECT brain radiotracer for the gonadotropin releasing hormone receptor

ανά Fjellaksel, Richard, Oteiza, Ana, Martin-Armas, Montserrat, Riss, Patrick J., Hjelstuen, Ole Kristian, Kuttner, Samuel, Hansen, Jørn H., Sundset, Rune
Τόπος έκδοσης BMC Res Notes (2018)

[(18)F]PR04.MZ PET/CT Imaging for Evaluation of Nigrostriatal Neuron Integrity in Patients With Parkinson Disease

ανά Juri, Carlos, Kramer, Vasko, Riss, Patrick J., Soza-Ried, Cristian, Haeger, Arlette, Pruzzo, Rossana, Rösch, Frank, Amaral, Horacio, Chana-Cuevas, Pedro
Τόπος έκδοσης Clin Nucl Med (2021)

Pharmacological Characterization of Low-to-Moderate Affinity Opioid Receptor Agonists and Brain Imaging with (18)F-Labeled Derivatives in Rats

ανά Ott, Julian, Spilhaug, Mona M., Maschauer, Simone, Rafique, Waqas, Jakobsson, Jimmy E., Hartvig, Karoline, Hübner, Harald, Gmeiner, Peter, Prante, Olaf, Riss, Patrick J.
Τόπος έκδοσης J Med Chem (2020)

Discovery of a Lead Brain‐Penetrating Gonadotropin‐Releasing Hormone Receptor Antagonist with Saturable Binding in Brain

ανά Bekker, Roberto B. W., Fjellaksel, Richard, Hjornevik, Trine, Nuruddin, Syed, Rafique, Waqas, Hansen, Jørn H., Sundset, Rune, Haraldsen, Ira H., Riss, Patrick J.
Τόπος έκδοσης ChemMedChem (2020)

Image-Guided Development of Heterocyclic Sulfoxides as Ligands for Tau Neurofibrillary Tangles: From First-in-Man to Second-Generation Ligands

ανά Rafique, Waqas, Kramer, Vasko, Pardo, Tania, Smits, René, Spilhaug, Mona M., Hoepping, Alexander, Savio, Eduardo, Engler, Henry, Kuljs, Rodrigo, Amaral, Horacio, Riss, Patrick J.
Τόπος έκδοσης ACS Omega (2018)

Validation and quantification of [(18)F]altanserin binding in the rat brain using blood input and reference tissue modeling

ανά Riss, Patrick J, Hong, Young T, Williamson, David, Caprioli, Daniele, Sitnikov, Sergey, Ferrari, Valentina, Sawiak, Steve J, Baron, Jean-Claude, Dalley, Jeffrey W, Fryer, Tim D, Aigbirhio, Franklin I
Έκδοση 2011

Evaluation of [(18)F]N-methyl-lansoprazole as a tau PET imaging agent in first-in-human studies

ανά Kramer, Vasko, Brooks, Allen F., Haeger, Arlette, Kuljis, Rodrigo, Rafique, Waqas, Koeppe, Robert A., Raffel, David M., Frey, Kirk A., Amaral, Horacio, Scott, Peter J. H., Riss, Patrick J.
Τόπος έκδοσης ACS Chem Neurosci (2020)

Insula serotonin 2A receptor binding and gene expression contribute to serotonin transporter polymorphism anxious phenotype in primates

ανά Santangelo, Andrea M., Sawiak, Steve J., Fryer, Tim, Hong, Young, Shiba, Yoshiro, Clarke, Hannah F., Riss, Patrick J., Ferrari, Valentina, Tait, Roger, Suckling, John, Aigbirhio, Franklin I., Roberts, Angela C.
Τόπος έκδοσης Proc Natl Acad Sci U S A (2019)

Synthesis and Initial in Vivo Studies with [(11)C]SB-216763: The First Radiolabeled Brain Penetrative Inhibitor of GSK-3

ανά Li, Lei, Shao, Xia, Cole, Erin L., Ohnmacht, Stephan A., Ferrari, Valentina, Hong, Young T., Williamson, David J., Fryer, Tim D., Quesada, Carole A., Sherman, Phillip, Riss, Patrick J., Scott, Peter J. H., Aigbirhio, Franklin I.
Τόπος έκδοσης ACS Med Chem Lett (2015)