A General Protocol for Cu-Mediated Fluoro-deamination: Sandmeyer Fluorination of Diverse Aromatic Substrates

af Pérez-García, R. Manuel, Grønnevik, Gaute, Riss, Patrick J.
Udgivet i Org Lett (2021)

Synthesis and Characterization in Rodent Brain of the Subtype-Selective NR2B NMDA Receptor Ligand [(11)C]Ro04-5595 as a Potential Radiotracer for Positron Emission Tomography

af Jakobsson, Jimmy E., Gourni, Eleni, Khanapur, Shivashankar, Brito, Beatriz, Riss, Patrick J.
Udgivet i ACS Omega (2019)

Cu(I)-catalyzed (11)C-carboxylation of boronic acid esters: a rapid and convenient entry to (11)C-labeled carboxylic acids, esters and amides

af Riss, Patrick J., Lu, Shuiyu, Telu, Sanjay, Aigbirhio, Franklin I., Pike, Victor W.
Udgivet 2012

Small molecule piperazinyl-benzimidazole antagonists of the gonadotropin-releasing hormone (GnRH) receptor

af Fjellaksel, Richard, Boomgaren, Marc, Sundset, Rune, Haraldsen, Ira H., Hansen, Jørn H., Riss, Patrick J.
Udgivet i Medchemcomm (2017)

Recent Development of Non-Peptide GnRH Antagonists

af Tukun, Feng-Ling, Olberg, Dag Erlend, Riss, Patrick J., Haraldsen, Ira, Kaass, Anita, Klaveness, Jo
Udgivet i Molecules (2017)

Radiosynthesis and validation of (18)F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain

af Cumming, Paul, Maschauer, Simone, Riss, Patrick J, Tschammer, Nuska, Fehler, Stefanie K, Heinrich, Markus R, Kuwert, Torsten, Prante, Olaf
Udgivet 2014

First in vivo evaluation of a potential SPECT brain radiotracer for the gonadotropin releasing hormone receptor

af Fjellaksel, Richard, Oteiza, Ana, Martin-Armas, Montserrat, Riss, Patrick J., Hjelstuen, Ole Kristian, Kuttner, Samuel, Hansen, Jørn H., Sundset, Rune
Udgivet i BMC Res Notes (2018)

[(18)F]PR04.MZ PET/CT Imaging for Evaluation of Nigrostriatal Neuron Integrity in Patients With Parkinson Disease

af Juri, Carlos, Kramer, Vasko, Riss, Patrick J., Soza-Ried, Cristian, Haeger, Arlette, Pruzzo, Rossana, Rösch, Frank, Amaral, Horacio, Chana-Cuevas, Pedro
Udgivet i Clin Nucl Med (2021)

Pharmacological Characterization of Low-to-Moderate Affinity Opioid Receptor Agonists and Brain Imaging with (18)F-Labeled Derivatives in Rats

af Ott, Julian, Spilhaug, Mona M., Maschauer, Simone, Rafique, Waqas, Jakobsson, Jimmy E., Hartvig, Karoline, Hübner, Harald, Gmeiner, Peter, Prante, Olaf, Riss, Patrick J.
Udgivet i J Med Chem (2020)

Discovery of a Lead Brain‐Penetrating Gonadotropin‐Releasing Hormone Receptor Antagonist with Saturable Binding in Brain

af Bekker, Roberto B. W., Fjellaksel, Richard, Hjornevik, Trine, Nuruddin, Syed, Rafique, Waqas, Hansen, Jørn H., Sundset, Rune, Haraldsen, Ira H., Riss, Patrick J.
Udgivet i ChemMedChem (2020)

Image-Guided Development of Heterocyclic Sulfoxides as Ligands for Tau Neurofibrillary Tangles: From First-in-Man to Second-Generation Ligands

af Rafique, Waqas, Kramer, Vasko, Pardo, Tania, Smits, René, Spilhaug, Mona M., Hoepping, Alexander, Savio, Eduardo, Engler, Henry, Kuljs, Rodrigo, Amaral, Horacio, Riss, Patrick J.
Udgivet i ACS Omega (2018)

Validation and quantification of [(18)F]altanserin binding in the rat brain using blood input and reference tissue modeling

af Riss, Patrick J, Hong, Young T, Williamson, David, Caprioli, Daniele, Sitnikov, Sergey, Ferrari, Valentina, Sawiak, Steve J, Baron, Jean-Claude, Dalley, Jeffrey W, Fryer, Tim D, Aigbirhio, Franklin I
Udgivet 2011

Evaluation of [(18)F]N-methyl-lansoprazole as a tau PET imaging agent in first-in-human studies

af Kramer, Vasko, Brooks, Allen F., Haeger, Arlette, Kuljis, Rodrigo, Rafique, Waqas, Koeppe, Robert A., Raffel, David M., Frey, Kirk A., Amaral, Horacio, Scott, Peter J. H., Riss, Patrick J.
Udgivet i ACS Chem Neurosci (2020)

Insula serotonin 2A receptor binding and gene expression contribute to serotonin transporter polymorphism anxious phenotype in primates

af Santangelo, Andrea M., Sawiak, Steve J., Fryer, Tim, Hong, Young, Shiba, Yoshiro, Clarke, Hannah F., Riss, Patrick J., Ferrari, Valentina, Tait, Roger, Suckling, John, Aigbirhio, Franklin I., Roberts, Angela C.
Udgivet i Proc Natl Acad Sci U S A (2019)

Synthesis and Initial in Vivo Studies with [(11)C]SB-216763: The First Radiolabeled Brain Penetrative Inhibitor of GSK-3

af Li, Lei, Shao, Xia, Cole, Erin L., Ohnmacht, Stephan A., Ferrari, Valentina, Hong, Young T., Williamson, David J., Fryer, Tim D., Quesada, Carole A., Sherman, Phillip, Riss, Patrick J., Scott, Peter J. H., Aigbirhio, Franklin I.
Udgivet i ACS Med Chem Lett (2015)