Enthalpy-Entropy Compensation in the Binding of Modulators at Ionotropic Glutamate Receptor GluA2

Por Krintel, Christian, Francotte, Pierre, Pickering, Darryl S., Juknaitė, Lina, Pøhlsgaard, Jacob, Olsen, Lars, Frydenvang, Karla, Goffin, Eric, Pirotte, Bernard, Kastrup, Jette S.
Publicado no Biophys J (2016)

Identification and pharmacological characterization of succinate receptor agonists

Por Geubelle, Pierre, Gilissen, Julie, Dilly, Sébastien, Poma, Laurence, Dupuis, Nadine, Laschet, Céline, Abboud, Dayana, Inoue, Asuka, Jouret, François, Pirotte, Bernard, Hanson, Julien
Publicado no Br J Pharmacol (2017)

Simple di- and trivanillates exhibit cytostatic properties toward cancer cells resistant to pro-apoptotic stimuli

Por Lamoral-Theys, Delphine, Pottier, Laurent, Kerff, Frédéric, Dufrasne, François, Proutière, Fabien, Wauthoz, Nathalie, Neven, Philippe, Ingrassia, Laurent, Van Antwerpen, Pierre, Lefranc, Florence, Gelbcke, Michel, Pirotte, Bernard, Kraus, Jean-Louis, Nève, Jean, Kornienko, Alexander, Kiss, Robert, Dubois, Jacques
Publicado no Bioorg Med Chem (2010)

7-Phenoxy-substituted 3,4-Dihydro-2H-1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors...

Por Goffin, Eric, Drapier, Thomas, Larsen, Anja Probst, Geubelle, Pierre, Ptak, Christopher P., Laulumaa, Saara, Rovinskaja, Karoline, Gilissen, Julie, de Tullio, Pascal, Olsen, Lars, Frydenvang, Karla, Pirotte, Bernard, Hanson, Julien, Oswald, Robert E., Kastrup, Jette Sandholm, Francotte, Pierre
Publicado no J Med Chem (2017)