Discovery of BMS-846372, a Potent and Orally Active Human CGRP Receptor Antagonist for the Treatment of Migraine

ανά Luo, Guanglin, Chen, Ling, Conway, Charles M., Denton, Rex, Keavy, Deborah, Gulianello, Michael, Huang, Yanling, Kostich, Walter, Lentz, Kimberley A., Mercer, Stephen E., Schartman, Richard, Signor, Laura, Browning, Marc, Macor, John E., Dubowchik, Gene M.
Έκδοση 2012

Development of 1H-Pyrazolo[3,4-b]pyridines as Metabotropic Glutamate Receptor 5 Positive Allosteric Modulators

ανά Hill, Matthew D., Fang, Haiquan, Brown, Jeffrey M., Molski, Thaddeus, Easton, Amy, Han, Xiaojun, Miller, Regina, Hill-Drzewi, Melissa, Gallagher, Lizbeth, Matchett, Michele, Gulianello, Michael, Balakrishnan, Anand, Bertekap, Robert L., Santone, Kenneth S., Whiterock, Valerie J., Zhuo, Xiaoliang, Bronson, Joanne J., Macor, John E., Degnan, Andrew P.
Τόπος έκδοσης ACS Med Chem Lett (2016)

Discovery and Preclinical Evaluation of BMS-955829, a Potent Positive Allosteric Modulator of mGluR5

ανά Yang, Fukang, Snyder, Lawrence B., Balakrishnan, Anand, Brown, Jeffrey M., Sivarao, Digavalli V., Easton, Amy, Fernandes, Alda, Gulianello, Michael, Hanumegowda, Umesh M., Huang, Hong, Huang, Yanling, Jones, Kelli M., Li, Yu-Wen, Matchett, Michele, Mattson, Gail, Miller, Regina, Santone, Kenneth S., Senapati, Arun, Shields, Eric E., Simutis, Frank J., Westphal, Ryan, Whiterock, Valerie J., Bronson, Joanne J., Macor, John E., Degnan, Andrew P.
Τόπος έκδοσης ACS Med Chem Lett (2016)

Inhibition of AAK1 Kinase as a Novel Therapeutic Approach to Treat Neuropathic Pain

ανά Kostich, Walter, Hamman, Brian D., Li, Yu-Wen, Naidu, Sreenivasulu, Dandapani, Kumaran, Feng, Jianlin, Easton, Amy, Bourin, Clotilde, Baker, Kevin, Allen, Jason, Savelieva, Katerina, Louis, Justin V., Dokania, Manoj, Elavazhagan, Saravanan, Vattikundala, Pradeep, Sharma, Vivek, Das, Manish Lal, Shankar, Ganesh, Kumar, Anoop, Holenarsipur, Vinay K., Gulianello, Michael, Molski, Ted, Brown, Jeffrey M., Lewis, Martin, Huang, Yanling, Lu, Yifeng, Pieschl, Rick, O’Malley, Kevin, Lippy, Jonathan, Nouraldeen, Amr, Lanthorn, Thomas H., Ye, Guilan, Wilson, Alan, Balakrishnan, Anand, Denton, Rex, Grace, James E., Lentz, Kimberley A., Santone, Kenneth S., Bi, Yingzhi, Main, Alan, Swaffield, Jon, Carson, Ken, Mandlekar, Sandhya, Vikramadithyan, Reeba K., Nara, Susheel J., Dzierba, Carolyn, Bronson, Joanne, Macor, John E., Zaczek, Robert, Westphal, Ryan, Kiss, Laszlo, Bristow, Linda, Conway, Charles M., Zambrowicz, Brian, Albright, Charles F.
Τόπος έκδοσης J Pharmacol Exp Ther (2016)