Synthesis and structure-activity relationships of a series 4-methoxy-3-(piperidin-4-yl)oxy benzamides as novel inhibitors of the presynaptic choline transporter

Por Bollinger, Sean R., Engers, Darren W., Ennis, Elizabeth A., Wright, Jane, Locuson, Charles W., Lindsley, Craig W., Blakely, Randy D., Hopkins, Corey R.
Publicado no Bioorg Med Chem Lett (2015)

Transgenic overexpression of the presynaptic choline transporter elevates acetylcholine levels and augments motor endurance

Por Holmstrand, Ericka C., Lund, David, Cherian, Ajeesh Koshy, Wright, Jane, Martin, Rolicia F., Ennis, Elizabeth A., Stanwood, Gregg D., Sarter, Martin, Blakely, Randy D.
Publicado em 2013

Nonoisotopic Assay for the Presynaptic Choline Transporter Reveals Capacity for Allosteric Modulation of Choline Uptake

Por Ruggiero, Alicia M., Wright, Jane, Ferguson, Shawn M., Lewis, Michelle, Emerson, Katie S., Iwamoto, Hideki, Ivy, Michael T., Holmstrand, Ericka C., Ennis, Elizabeth. A., Weaver, C. David, Blakely, Randy D.
Publicado em 2012

Identification and Characterization of ML352: A Novel, Noncompetitive Inhibitor of the Presynaptic Choline Transporter

Por Ennis, Elizabeth A., Wright, Jane, Retzlaff, Cassandra L., McManus, Owen B., Lin, Zhinong, Huang, Xiaofang, Wu, Meng, Li, Min, Daniels, J. Scott, Lindsley, Craig W., Hopkins, Corey R., Blakely, Randy D.
Publicado no ACS Chem Neurosci (2015)