Discovery of N-[4-(1H-Pyrazolo[3,4-b]pyrazin-6-yl)-phenyl]-sulfonamides as Highly Active and Selective SGK1 Inhibitors

по Halland, Nis, Schmidt, Friedemann, Weiss, Tilo, Saas, Joachim, Li, Ziyu, Czech, Jörg, Dreyer, Matthias, Hofmeister, Armin, Mertsch, Katharina, Dietz, Uwe, Strübing, Carsten, Nazare, Marc
Опубликовано в: ACS Med Chem Lett (2014)

Isolation, Co-Crystallization and Structure-Based Characterization of Anabaenopeptins as Highly Potent Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (TAFIa)

по Schreuder, Herman, Liesum, Alexander, Lönze, Petra, Stump, Heike, Hoffmann, Holger, Schiell, Matthias, Kurz, Michael, Toti, Luigi, Bauer, Armin, Kallus, Christopher, Klemke-Jahn, Christine, Czech, Jörg, Kramer, Dan, Enke, Heike, Niedermeyer, Timo H. J., Morrison, Vincent, Kumar, Vasant, Brönstrup, Mark
Опубликовано в: Sci Rep (2016)

Activation of Adenosine Monophosphate—Activated Protein Kinase Reduces the Onset of Diet‐Induced Hepatocellular Carcinoma in Mice

по Schmoll, Dieter, Ziegler, Nicole, Viollet, Benoit, Foretz, Marc, Even, Patrick C., Azzout‐Marniche, Dalila, Nygaard Madsen, Andreas, Illemann, Martin, Mandrup, Karen, Feigh, Michael, Czech, Jörg, Glombik, Heiner, Olsen, Jacob A., Hennerici, Wolfgang, Steinmeyer, Klaus, Elvert, Ralf, Castañeda, Tamara R., Kannt, Aimo
Опубликовано в: Hepatol Commun (2020)

A small molecule inhibitor of Nicotinamide N-methyltransferase for the treatment of metabolic disorders

по Kannt, Aimo, Rajagopal, Sridharan, Kadnur, Sanjay Venkatachalapathi, Suresh, Juluri, Bhamidipati, Ravi Kanth, Swaminathan, Srinivasan, Hallur, Mahanandeesha Siddappa, Kristam, Rajendra, Elvert, Ralf, Czech, Jörg, Pfenninger, Anja, Rudolph, Christine, Schreuder, Herman, Chandrasekar, Devaraj Venkatapura, Mane, Vishal Subhash, Birudukota, Swarnakumari, Shaik, Shama, Zope, Bharat Ravindra, Burri, Raghunadha Reddy, Anand, Niranjan Naranapura, Thakur, Manish Kumar, Singh, Manvi, Parveen, Reejuana, Kandan, Saravanan, Mullangi, Ramesh, Yura, Takeshi, Gosu, Ramachandraiah, Ruf, Sven, Dhakshinamoorthy, Saravanakumar
Опубликовано в: Sci Rep (2018)