Design, Synthesis, Docking Studies and Monoamine Oxidase Inhibition of a Small Library of 1-acetyl- and 1-thiocarbamoyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazoles

por Guglielmi, Paolo, Carradori, Simone, Poli, Giulio, Secci, Daniela, Cirilli, Roberto, Rotondi, Giulia, Chimenti, Paola, Petzer, Anél, Petzer, Jacobus P.
Publicado en Molecules (2019)

Novel insights on saccharin- and acesulfame-based carbonic anhydrase inhibitors: design, synthesis, modelling investigations and biological activity evaluation

por Guglielmi, Paolo, Rotondi, Giulia, Secci, Daniela, Angeli, Andrea, Chimenti, Paola, Nocentini, Alessio, Bonardi, Alessandro, Gratteri, Paola, Carradori, Simone, Supuran, Claudiu T.
Publicado en J Enzyme Inhib Med Chem (2020)

Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives

por Carradori, Simone, Secci, Daniela, Bizzarri, Bruna, Chimenti, Paola, De Monte, Celeste, Guglielmi, Paolo, Campestre, Cristina, Rivanera, Daniela, Bordón, Claudia, Jones-Brando, Lorraine
Publicado en J Enzyme Inhib Med Chem (2017)

4-(3-Nitrophenyl)thiazol-2-ylhydrazone derivatives as antioxidants and selective hMAO-B inhibitors: synthesis, biological activity and computational analysis

por Secci, Daniela, Carradori, Simone, Petzer, Anél, Guglielmi, Paolo, D’Ascenzio, Melissa, Chimenti, Paola, Bagetta, Donatella, Alcaro, Stefano, Zengin, Gokhan, Petzer, Jacobus P., Ortuso, Francesco
Publicado en J Enzyme Inhib Med Chem (2019)

Benzo[b]tiophen-3-ol derivatives as effective inhibitors of human monoamine oxidase: design, synthesis, and biological activity

por Guglielmi, Paolo, Secci, Daniela, Petzer, Anél, Bagetta, Donatella, Chimenti, Paola, Rotondi, Giulia, Ferrante, Claudio, Recinella, Lucia, Leone, Sheila, Alcaro, Stefano, Zengin, Gokhan, Petzer, Jacobus P., Ortuso, Francesco, Carradori, Simone
Publicado en J Enzyme Inhib Med Chem (2019)