Multiple N-methylation of MT-II backbone amide bonds leads to melanocortin receptor subtype hMC1R selectivity; pharmacological and conformational studies

由 Doedens, Lucas, Opperer, Florian, Cai, Minying, Beck, Johannes G., Dedek, Matt, Palmer, Erin, Hruby, Victor J., Kessler, Horst
出版 2010

Structural Insights into Selective Ligand–Receptor Interactions Leading to Receptor Inactivation Utilizing Selective Melanocortin 3 Receptor Antagonists

由 Cai, Minying, Marelli, Udaya Kiran, Mertz, Blake, Beck, Johannes G., Opperer, Florian, Rechenmacher, Florian, Kessler, Horst, Hruby, Victor J.
發表在 Biochemistry (2017)

N-Methylated sst(2) Selective Somatostatin Cyclic Peptide Analogue as a Potent Candidate for Treating Neurogenic Inflammation

由 Chatterjee, Jayanta, Laufer, Burkhardt, Beck, Johannes G., Helyes, Zsuzsanna, Pintér, Erika, Szolcsányi, János, Horvath, Aniko, Mandl, Jozsef, Reubi, Jean C., Kéri, György, Kessler, Horst
出版 2011

Systematic Backbone Conformational Constraints on a Cyclic Melanotropin Ligand Leads to Highly Selective Ligands for Multiple Melanocortin Receptors

由 Cai, Minying, Marelli, Udaya Kiran, Bao, Jennifer, Beck, Johannes G., Opperer, Florian, Rechenmacher, Florian, McLeod, Kaitlyn R., Zingsheim, Morgan R., Doedens, Lucas, Kessler, Horst, Hruby, Victor J.
發表在 J Med Chem (2015)