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Timing of Novel Drug 1A-116 to Circadian Rhythms Improves Therapeutic Effects against Glioblastoma

The Ras homologous family of small guanosine triphosphate-binding enzymes (GTPases) is critical for cell migration and proliferation. The novel drug 1A-116 blocks the interaction site of the Ras-related C3 botulinum toxin substrate 1 (RAC1) GTPase with some of its guanine exchange factors (GEFs), su...

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Publicat a:Pharmaceutics
Autors principals: Trebucq, Laura Lucía, Cardama, Georgina Alexandra, Lorenzano Menna, Pablo, Golombek, Diego Andrés, Chiesa, Juan José, Marpegan, Luciano
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC8309043/
https://ncbi.nlm.nih.gov/pubmed/34371781
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics13071091
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