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Exploring the chemical space of protein–protein interaction inhibitors through machine learning

Although protein–protein interactions (PPIs) have emerged as the basis of potential new therapeutic approaches, targeting intracellular PPIs with small molecule inhibitors is conventionally considered highly challenging. Driven by increasing research efforts, success rates have increased significant...

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Dettagli Bibliografici
Pubblicato in:Sci Rep
Autori principali: Choi, Jiwon, Yun, Jun Seop, Song, Hyeeun, Kim, Nam Hee, Kim, Hyun Sil, Yook, Jong In
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group UK 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8238997/
https://ncbi.nlm.nih.gov/pubmed/34183730
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-021-92825-5
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