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Ring-fused cyclobutanes via cycloisomerization of alkylidenecyclopropane acylsilanes

A novel Lewis acid-catalyzed cycloisomerization of alkylidenecyclopropane acylsilanes is disclosed. The readily available starting materials participate in tandem Prins addition/ring expansion/1,2-silyl shift to grant access to bicyclo[4.2.0]octanes and bicyclo[3.2.0]heptanes, which are common motif...

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Detalhes bibliográficos
Publicado no:Chem Sci
Main Authors: Eichenberger, Sarah, Hönig, Moritz, Richter, Matthieu J. R., Gershoni-Poranne, Renana, Carreira, Erick M.
Formato: Artigo
Idioma:Inglês
Publicado em: The Royal Society of Chemistry 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC8159344/
https://ncbi.nlm.nih.gov/pubmed/34122987
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0sc02224a
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