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(177)Lu-Labeled Albumin-Binder–Conjugated PSMA-Targeting Agents with Extremely High Tumor Uptake and Enhanced Tumor-to-Kidney Absorbed Dose Ratio

The use of an albumin binder has been shown to improve tumor uptake of prostate-specific membrane antigen (PSMA)–targeting radiotherapeutic agents. The aim of this study was to develop improved radiotherapeutic agents that combine an optimized affinity-modifying group and optimized albumin binders t...

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Pubblicato in:J Nucl Med
Autori principali: Kuo, Hsiou-Ting, Lin, Kuo-Shyan, Zhang, Zhengxing, Uribe, Carlos F., Merkens, Helen, Zhang, Chengcheng, Bénard, François
Natura: Artigo
Lingua:Inglês
Pubblicazione: Society of Nuclear Medicine 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC8049373/
https://ncbi.nlm.nih.gov/pubmed/32859704
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.2967/jnumed.120.250738
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