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In silico investigation of potential small molecule inhibitors of the SARS-CoV-2 nsp10-nsp16 methyltransferase complex

The COVID-19 pandemic caused by SARS-CoV-2 has resulted in an international health emergency. The SARS-CoV-2 nsp16 is an S-adenosyl-L-methionine (SAM)-dependent methyltransferase, and with its cofactor nsp10, is responsible for RNA cap formation. This study aimed to identify small molecules binding...

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Publicado en:Chem Phys Lett
Autores principales: Liang, Julia, Pitsillou, Eleni, Burbury, Lucy, Hung, Andrew, Karagiannis, Tom C.
Formato: Artigo
Lenguaje:Inglês
Publicado: Elsevier B.V. 2021
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC8032478/
https://ncbi.nlm.nih.gov/pubmed/33850334
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.cplett.2021.138618
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