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Resistance to BET inhibitors in lung adenocarcinoma is mediated by casein kinase phosphorylation of BRD4

Targeting the epigenome to modulate gene expression programs driving cancer development has emerged as an exciting avenue for therapeutic intervention. Pharmacological inhibition of the bromodomain and extraterminal (BET) family of chromatin adapter proteins has proven effective in this regard, supp...

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Pubblicato in:Oncogenesis
Autori principali: Calder, Jack, Nagelberg, Amy, Luu, Jennifer, Lu, Daniel, Lockwood, William W.
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group UK 2021
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7955060/
https://ncbi.nlm.nih.gov/pubmed/33712563
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41389-021-00316-z
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