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Clinical Pharmacokinetics and Pharmacodynamics of Selumetinib

Selumetinib, a highly specific MEK1/2 inhibitor, is approved for children older than 2 years of age with neurofibromatosis 1 (NF1) who have inoperable plexiform neurofibromas. By selectively binding to MEK1/2 proteins, selumetinib can arrest the mitogen-activated protein kinases/extracellular signal...

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Pubblicato in:Clin Pharmacokinet
Autori principali: Campagne, Olivia, Yeo, Kee Kiat, Fangusaro, Jason, Stewart, Clinton F.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7935771/
https://ncbi.nlm.nih.gov/pubmed/33354735
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s40262-020-00967-y
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