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Discovery of a Positron Emission Tomography Radiotracer Selectively Targeting the BD1 Bromodomains of BET Proteins
[Image: see text] In this paper, we report the design, synthesis, and biological evaluation of the first selective bromodomain and extra-terminal domain (BET) BD1 bromodomains of the PET radiotracer [(18)F]PB006. The standard compound PB006 showed high affinity and good selectivity toward BRD4 BD1 (...
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| Publicat a: | ACS Med Chem Lett |
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| Autors principals: | , , , , , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
American Chemical Society
2021
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| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7883468/ https://ncbi.nlm.nih.gov/pubmed/33603976 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.0c00650 |
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