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Potency Increase of Spiroketal Analogs of Membrane Inserting Indolyl Mannich Base Antimycobacterials Is Due to Acquisition of MmpL3 Inhibition

Chemistry campaigns identified amphiphilic indolyl Mannich bases as novel membrane-permeabilizing antimycobacterials. Spiroketal analogs of this series showed increased potency and the lead compound 1 displayed efficacy in a mouse model of tuberculosis. Yet the mechanism by which the spiroketal moie...

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Detalhes bibliográficos
Publicado no:ACS Infect Dis
Main Authors: Li, Ming, Phua, Zheng Yen, Xi, Yu, Xu, Zhujun, Nyantakyi, Samuel A., Li, Wei, Jackson, Mary, Wong, Ming Wah, Lam, Yulin, Chng, Shu Sin, Go, Mei Lin, Dick, Thomas
Formato: Artigo
Idioma:Inglês
Publicado em: 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7875313/
https://ncbi.nlm.nih.gov/pubmed/32413266
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsinfecdis.0c00121
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