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BMI1-Inhibitor PTC596 in Combination with MCL1 Inhibitor S63845 or MEK Inhibitor Trametinib in the Treatment of Acute Leukemia

SIMPLE SUMMARY: Prognosis for acute myeloid leukemia (AML) patients is poor, particularly in TP53 mutated AML, secondary, relapsed, and refractory AML, and in patients unfit for intensive treatment, thus highlighting an unmet need for novel therapeutic approaches. Targeting the stem cell oncoprotein...

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Publicado en:Cancers (Basel)
Autores principales: Seipel, Katja, Kopp, Basil, Bacher, Ulrike, Pabst, Thomas
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI 2021
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7867282/
https://ncbi.nlm.nih.gov/pubmed/33540760
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/cancers13030581
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