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Analyzing Kinase Similarity in Small Molecule and Protein Structural Space to Explore the Limits of Multi-Target Screening

While selective inhibition is one of the key assets for a small molecule drug, many diseases can only be tackled by simultaneous inhibition of several proteins. An example where achieving selectivity is especially challenging are ligands targeting human kinases. This difficulty arises from the high...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Molecules
Hauptverfasser: Schmidt, Denis, Scharf, Magdalena M., Sydow, Dominique, Aßmann, Eva, Martí-Solano, Maria, Keul, Marina, Volkamer, Andrea, Kolb, Peter
Format: Artigo
Sprache:Inglês
Veröffentlicht: MDPI 2021
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7865522/
https://ncbi.nlm.nih.gov/pubmed/33530327
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules26030629
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