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Inclusion Compound of Efavirenz and γ-Cyclodextrin: Solid State Studies and Effect on Solubility

Efavirenz is an antiretroviral drug of widespread use in the management of infections with human immunodeficiency virus type 1 (HIV-1). Efavirenz is also used in paediatrics, but due to its very poor aqueous solubility the liquid formulations available resort to oil-based excipients. In this report...

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Publicat a:Molecules
Autors principals: Braga, Susana Santos, El-Saleh, Firas, Lysenko, Karyna, Paz, Filipe A. Almeida
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2021
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7863942/
https://ncbi.nlm.nih.gov/pubmed/33498239
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules26030519
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