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Protocol for hit-to-lead optimization of compounds by auto in silico ligand directing evolution (AILDE) approach
Hit-to-lead (H2L) optimization is crucial for drug design, which has become an increasing concern in medicinal chemistry. A virtual screening strategy of auto in silico ligand directing evolution (AILDE) has been developed to yield promising lead compounds rapidly and efficiently. The protocol inclu...
Αποθηκεύτηκε σε:
| Τόπος έκδοσης: | STAR Protoc |
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| Κύριοι συγγραφείς: | , , , |
| Μορφή: | Artigo |
| Γλώσσα: | Inglês |
| Έκδοση: |
Elsevier
2021
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| Θέματα: | |
| Διαθέσιμο Online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7856476/ https://ncbi.nlm.nih.gov/pubmed/33554146 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.xpro.2021.100312 |
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