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Synthesis and Antiplasmodial Activity of Novel Bioinspired Imidazolidinedione Derivatives

Malaria is an enormous threat to public health, due to the emergence of Plasmodium falciparum resistance to widely-used antimalarials, such as chloroquine (CQ). Current antimalarial drugs are aromatic heterocyclic derivatives, most often containing a basic component with an added alkyl chain in thei...

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Vydáno v:Biomolecules
Hlavní autoři: Jaromin, Anna, Czopek, Anna, Parapini, Silvia, Basilico, Nicoletta, Misiak, Ernest, Gubernator, Jerzy, Zagórska, Agnieszka
Médium: Artigo
Jazyk:Inglês
Vydáno: MDPI 2020
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7823712/
https://ncbi.nlm.nih.gov/pubmed/33383906
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biom11010033
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