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Activity and bioavailability of tepotinib for leptomeningeal metastasis of NSCLC with MET exon 14 skipping mutation

Tepotinib is a key drug for cancer patients with mesenchymal‐epithelial transition receptor tyrosine kinase proto‐oncogene (MET) exon 14 skipping mutation. However, its bioavailability in the cerebrospinal fluid (CSF) in humans has not been fully elucidated. Moreover, information about the efficacy...

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Dettagli Bibliografici
Pubblicato in:Cancer Commun (Lond)
Autori principali: Tanaka, Hisashi, Taima, Kageaki, Makiguchi, Tomonori, Nakagawa, Junichi, Niioka, Takenori, Tasaka, Sadatomo
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley and Sons Inc. 2021
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7819565/
https://ncbi.nlm.nih.gov/pubmed/33387444
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cac2.12124
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