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Using machine learning to improve ensemble docking for drug discovery

Ensemble docking has provided an inexpensive method to account for receptor flexibility in molecular docking for virtual screening. Unfortunately, as there is no rigorous theory to connect the docking scores from multiple structures to measured activity, researchers have not yet come up with effecti...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Proteins
Egile Nagusiak: Chandak, Tanay, Mayginnes, John P., Mayes, Howard, Wong, Chung F.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2020
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC7815257/
https://ncbi.nlm.nih.gov/pubmed/32401384
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prot.25899
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