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Molecular Simulation and Statistical Learning Methods toward Predicting Drug–Polymer Amorphous Solid Dispersion Miscibility, Stability, and Formulation Design

Amorphous solid dispersions (ASDs) have emerged as widespread formulations for drug delivery of poorly soluble active pharmaceutical ingredients (APIs). Predicting the API solubility with various carriers in the API–carrier mixture and the principal API–carrier non-bonding interactions are critical...

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Dettagli Bibliografici
Pubblicato in:Molecules
Autori principali: Walden, Daniel M., Bundey, Yogesh, Jagarapu, Aditya, Antontsev, Victor, Chakravarty, Kaushik, Varshney, Jyotika
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2021
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7794704/
https://ncbi.nlm.nih.gov/pubmed/33401494
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules26010182
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