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Identification of Enzymes Oxidizing the Tyrosine Kinase Inhibitor Cabozantinib: Cabozantinib Is Predominantly Oxidized by CYP3A4 and Its Oxidation Is Stimulated by cyt b(5) Activity

Herein, the in vitro metabolism of tyrosine kinase inhibitor cabozantinib, the drug used for the treatment of metastatic medullary thyroid cancer and advanced renal cell carcinoma, was studied using hepatic microsomal samples of different human donors, human recombinant cytochromes P450 (CYPs), flav...

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Detalhes bibliográficos
Publicado no:Biomedicines
Main Authors: Indra, Radek, Vavrová, Katarína, Pompach, Petr, Heger, Zbyněk, Hodek, Petr
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7759869/
https://ncbi.nlm.nih.gov/pubmed/33260548
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/biomedicines8120547
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