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Target-Mediated Brain Tissue Binding for Small Molecule Inhibitors of Heat Shock Protein 90

Drug distribution in the brain is generally associated with an affinity for fatty brain tissues and therefore known to be species- and concentration-independent. We report here the effect of target affinity on brain tissue binding for 10 small molecules designed to inhibit brain heat shock protein 9...

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Dettagli Bibliografici
Pubblicato in:Pharmaceutics
Autori principali: Badolo, Lassina, Thirstrup, Kenneth, Nielsen, Søren Møller, Püschl, Ask, Jensen, Thomas, Watson, Steve, Bundgaard, Christoffer
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7690585/
https://ncbi.nlm.nih.gov/pubmed/33105895
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/pharmaceutics12111009
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