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DRUG MIMICRY: PROMISCUOUS RECEPTORS PXR and AhR AND MICROBIAL METABOLITE INTERACTIONS IN THE INTESTINE

Significant attrition limits drug discovery. The available chemical entities present with drug-like features contribute to this limitation. Using specific examples of promiscuous receptor-ligand interactions, we make a case for expanding the chemical space for drug-like molecules. These ligand-recep...

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Détails bibliographiques
Publié dans:Trends Pharmacol Sci
Auteurs principaux: Dvořák, Zdeněk, Sokol, Harry, Mani, Sridhar
Format: Artigo
Langue:Inglês
Publié: 2020
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC7669654/
https://ncbi.nlm.nih.gov/pubmed/33097284
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tips.2020.09.013
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