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LigGrep: a tool for filtering docked poses to improve virtual-screening hit rates

Structure-based virtual screening (VS) uses computer docking to prioritize candidate small-molecule ligands for subsequent experimental testing. Docking programs evaluate molecular binding in part by predicting the geometry with which a given compound might bind a target receptor (e.g., the docked “...

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Publicat a:J Cheminform
Autors principals: Ha, Emily J., Lwin, Cara T., Durrant, Jacob D.
Format: Artigo
Idioma:Inglês
Publicat: Springer International Publishing 2020
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7656723/
https://ncbi.nlm.nih.gov/pubmed/33292486
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/s13321-020-00471-2
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